Association·arcadia

Mechanism of 48/80 toxicity is unrelated to MRGPRX2

Claim that 48/80’s toxicity is not caused by its canonical MRGPRX2 agonist activity but by some other, as-yet-unknown mechanism.

Confidence
80%
active

Evidence Quote

48/80 toxicity is not the direct result of MRGPRX2 activation but rather of some other as-yet-undescribed effect.

Relationship

toxicity hmc1.2 rbl2h3 not due to MRGPRX2 receptor

Evidence

Reference to the study examining genistein's inhibition of MRGPRX2 in relation to 48/80-induced anaphylactoid shock.

(2020). Protective Effect of Genistein against Compound 48/80 Induced Anaphylactoid Shock via Inhibiting MAS Related G Protein-Coupled Receptor X2 (MRGPRX2). doi:10.3390/molecules25051028